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AM-630– synthetic, CB2 antagonist

AM-630– synthetic, CB2 antagonist


AM630, a competitive cannabinoid receptor antagonist.      (abst – 1995)


Cannabinoid CB2 receptor activation reduces mouse myocardial ischemia-reperfusion injury: involvement of cytokine/chemokines and PMN                    (full – 2003)  cannabinoid&searchid=1&FIRSTINDEX=320&resourcetype=HWCIT


Inhibition of Inflammatory Hyperalgesia by Activation of Peripheral CB2 Cannabinoid Receptors                          (full – 2003)



Antinociceptive effect of cannabinoid agonist WIN 55,212–2 in rats with a spinal cord injury    (full – 2006)


Inhibition of Salivary Secretion by Activation of Cannabinoid Receptors       (full – 2006)       full   text=cannabinoid&searchid=1&FIRSTINDEX=880&resourcetype=HWCIT


The local antinociceptive effects of paracetamol in neuropathic pain are mediated by cannabinoid receptors                             (abst – 2007)


Regulation of Bone Mass, Osteoclast Function, and Ovariectomy-Induced Bone Loss by the Type 2 Cannabinoid Receptor                           (full – 2008)  ulltext=cannabinoid&searchid=1&FIRSTINDEX=240&resourcetype=HWCIT


Attenuation of Experimental Autoimmune Hepatitis by Exogenous and Endogenous Cannabinoids: Involvement of Regulatory T Cells                                 (full – 2008) ext=cannabinoid&searchid=1&FIRSTINDEX=320&resourcetype=HWCIT#content-block



Cannabinoid CB2 Receptor Potentiates Obesity-Associated Inflammation, Insulin Resistance and Hepatic Steatosis                                  (full – 2009)


Cannabinoid receptor-dependent and -independent anti-proliferative effects of omega-3 ethanolamides in androgen receptor-positive and -negative prostate cancer cell lines. (full – 2010)                     


A nonsynonymous polymorphism in cannabinoid CB2 receptor gene is associated with eating disorders in humans and food intake is modified in mice by its ligands.

(abst – 2010)


Cannabinoid receptor-2 (CB2) agonist ameliorates colitis in IL-10(-/-) mice by attenuating the activation of T cells and promoting their apoptosis.                                                  (abst – 2011)


Cannabinoid-2 Receptor Activation Protects against Infarct and Ischemia/Reperfusion Heart Injury.                            (abst – 2011)


The role of central CB2 cannabinoid receptors on food intake in neonatal chicks (abst – 2011)                 


Effects of a Selective Cannabinoid CB2 Agonist and Antagonist on Intravenous Nicotine Self Administration and Reinstatement of Nicotine Seeking.             (full – 2012)


Early Endogenous Activation of CB1 and CB2 Receptors after Spinal Cord Injury Is a Protective Response Involved in Spontaneous Recovery                        (full – 2012)


The role of CB2 receptor ligands in human eosinophil function     (full – 2012)


Effect of omega-3 polyunsaturated fatty acids on the endocannabinoid system in osteoblast-like cells and muscle                                         (abst – 2012)


Cannabinoids and muscular pain. Effectiveness of the local administration in rat. (abst – 2012)                   


Cannabinoids ameliorate disease progression in a model of multiple sclerosis in mice, acting preferentially through CB(1) receptor-mediated anti-inflammatory effects. (abst – 2012)                   


Cannabinoid receptor 2 agonist ameliorates mesenteric angiogenesis and portosystemic collaterals in cirrhotic rats.                            (abst – 2012)


Peripheral antinociceptive effect of anandamide and drugs that affect the endocannabinoid system on the formalin test in normal and streptozotocin-diabetic rats. (abst – 2012)                   


The maintenance of cisplatin- and paclitaxel-induced mechanical and cold allodynia is suppressed by cannabinoid CB2 receptor activation and independent of CXCR4 signaling in models of chemotherapy-induced peripheral neuropathy.                                                    (abst – 2012)


Anandamide enhances expression of heat shock protein 72 to protect against ischemia- reperfusion injury in rat heart.                                   (abst – 2012)


Diuretic effects of cannabinoids.  (abst – 2012)


Acute toxicity due to the confirmed consumption of synthetic cannabinoids: clinical and laboratory findings                            (abst – 2012)


Anti-Inflammatory Effect of the Endocannabinoid Anandamide in Experimental Periodontitis and Stress in the Rat                           (abst – 2012)


CB1 and CB2 Cannabinoid Receptor Agonists Induce Peripheral Antinociception by Activation of the Endogenous Noradrenergic System.                           (abst – 2013)


Inhibition of endocannabinoid degradation in experimental endotoxemia reduces leukocyte adhesion and improves capillary perfusion in the gut.                           (abst – 2013)


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