AM -2233 – synthetic, CB1 agonist

 

F200A substitution in the third transmembrane helix of human cannabinoid CB1 receptor converts AM2233 from receptor agonist to inverse agonist.                     (abst – 2006)  http://www.ncbi.nlm.nih.gov/pubmed/16438957

 

Evaluation of the in vivo receptor occupancy for the behavioral effects of cannabinoids using a radiolabeled cannabinoid receptor agonist, R-[125/131I]AM2233.

(abst – 2006)       http://www.ncbi.nlm.nih.gov/pubmed/16715483

 

Another nail in coffin of synthetic cannabis       (news – 2011)

http://tvnz.co.nz/national-news/another-nail-in-coffin-synthetic-cannabis-4666168?ref=rss

 

 

 

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