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ACEA/ ARACHIDONYL-2′-CHLOROETHYLAMIDE

ACEA/ARACHIDONYL-2′-CHLOROETHYLAMIDE– synthetic, CB1 agonist

 

Synthesis and characterization of potent and selective agonists of the neuronal cannabinoid receptor (CB1). (full – 1999) http://jpet.aspetjournals.org/content/289/3/1427.long

 

The cannabinoids R(-)-7-hydroxy-delta-6-tetra-hydrocannabinol-dimethylheptyl (HU- 210), 2-O-arachidonoylglycerylether (HU-310) and arachidonyl-2-chloroethylamide (ACEA) increase isoflurane provoked sleep duration by activation of cannabinoids 1 (CB1)-receptors in mice.     (abst – 2002)                                                           http://www.ncbi.nlm.nih.gov/pubmed/12095655

 

In vivo effects of CB1 receptor ligands on lipid peroxidation and antioxidant defense systems in the rat brain of healthy and ethanol-treated rats.                                                               (full – 2006)  http://www.if-pan.krakow.pl/pjp/pdf/2006/6_876.pdf

 

Differential effect of cannabinoid agonists and endocannabinoids on histamine release from distinct regions of the rat brain.                                                                  (full – 2006)  http://www.ncbi.nlm.nih.gov/pmc/articles/PMC1769340/?tool=pubmed

 

Arachidonyl-2′-chloroethylamide, a highly selective cannabinoid CB1 receptor agonist, enhances the anticonvulsant action of valproate in the mouse maximal electroshock- induced seizure model.     (abst – 2006)                                                         http://www.ncbi.nlm.nih.gov/pubmed/16930590

 

Opposing control of cannabinoid receptor stimulation on amyloid-beta-induced reactive gliosis: in vitro and in vivo evidence.                                                                  (full – 2007)  http://jpet.aspetjournals.org/content/322/3/1144.long

 

Ultra-low dose cannabinoid antagonist AM251 enhances cannabinoid anticonvulsant effects in the pentylenetetrazole-induced seizure in mice.                                            (abst – 2007)  http://www.ncbi.nlm.nih.gov/pubmed/17870135

 

Attenuation of Experimental Autoimmune Hepatitis by Exogenous and Endogenous Cannabinoids: Involvement of Regulatory T Cells                                                                        (full – 2008)  http://molpharm.aspetjournals.org/content/74/1/20.full?maxtoshow=&hits=80&RESULTFORMAT=&fullt  ext=cannabinoid&searchid=1&FIRSTINDEX=320&resourcetype=HWCIT#content-block

 

Cannabinoid modulation of cutaneous Adelta nociceptors during inflammation. (full – 2008)                                         http://www.ncbi.nlm.nih.gov/pmc/articles/PMC2585399/?tool=pubmed

 

Cannabinoid-mediated antinociception is enhanced in rat osteoarthritic knees. (full – 2008)                                         http://onlinelibrary.wiley.com/doi/10.1002/art.23156/full

 

Cannabinoid receptor activation induces apoptosis through tumor necrosis factor alpha- mediated ceramide de novo synthesis in colon cancer cells.                                                            (full – 2008)  http://clincancerres.aacrjournals.org/content/14/23/7691.long

 

Additive Interaction of the Cannabinoid Receptor I Agonist Arachidonyl-2- chloroethylamide with Etomidate in a Sedation Model in Mice                                                                           (full – 2008)  http://journals.lww.com/anesthesiology/Fulltext/2008/04000/Additive_Interaction_of_the_Cannabinoid_Re  ceptor_I.19.aspx

 

Peripheral cannabinoid CB1 receptors inhibit evoked responses of nociceptive neurones in vivo   (abst – 2008)                            http://www.sciencedirect.com/science/article/pii/S0014299908002719

 

Endogenous cannabinoids induce fever through the activation of CB1 receptors. (full – 2009)                                    http://www.ncbi.nlm.nih.gov/pmc/articles/PMC2765314/?tool=pubmed

 

The effects of intracerebroventricular AM-251, a CB1-receptor antagonist, and ACEA, a CB1-receptor agonist, on penicillin-induced epileptiform activity in rats.                                                         (full – 2009)  http://onlinelibrary.wiley.com/doi/10.1111/j.1528-1167.2009.02098.x/full

 

Involvement of nitrergic system in the anticonvulsant effect of the cannabinoid CB(1) agonist ACEA in the pentylenetetrazole-induced seizure in mice.                                                 (abst – 2009)  http://www.ncbi.nlm.nih.gov/pubmed/19223154

 

Involvement of nitric oxide in the gastroprotective effect of ACEA, a selective cannabinoid CB1 receptor agonist, on aspirin-induced gastric ulceration.                                                                      (abst – 2009)  http://www.ncbi.nlm.nih.gov/pubmed/19827302

 

Effect of arachidonyl-2′-chloroethylamide, a selective cannabinoid CB1 receptor agonist, on the protective action of the various antiepileptic drugs in the mouse maximal electroshock-induced seizure model.        (abst – 2009)  http://www.ncbi.nlm.nih.gov/pubmed/19751793

 

Role of cannabinoid CB1 receptors on macronutrient selection and satiety in rats. (abst – 2009)                                   http://www.ncbi.nlm.nih.gov/pubmed/19150453

 

Regulatory Role of Cannabinoid Receptor 1 in Stress-Induced Excitotoxicity and Neuroinflammation    (full – 2010)  http://www.nature.com/npp/journal/vaop/ncurrent/full/npp2010214a.html

 

Alkamides and a neolignan from Echinacea purpurea roots and the interaction of alkamides with G-protein-coupled cannabinoid receptors.                                                                       (abst – 2011)  http://www.ncbi.nlm.nih.gov/pubmed/21764086

 

The Effect of Hypoxia on G Protein Coupled (CB1) Receptor Gene Expression in Cortical B50 Neurons in Culture                                                                   (abst – 2011)  http://www.maxwellsci.com/jp/abstract.php?jid=BJPT&no=92&abs=05

 

Inhibition of basal and ultraviolet B-induced melanogenesis by cannabinoid CB(1) receptors: a keratinocyte-dependent effect.                                                       (abst – 2011)  http://www.ncbi.nlm.nih.gov/pubmed/21298280

 

L-Type Calcium Channel Mediates Anticonvulsant Effect of Cannabinoids in Acute and Chronic Murine Models of Seizure.                                                          (abst – 2011)  http://www.ncbi.nlm.nih.gov/pubmed/21928146

 

Changes in the cannabinoid (CB1) receptor expression level and G-protein activation in kainic acid induced seizures.                                            (abst – 2011)     http://www.ncbi.nlm.nih.gov/pubmed/22079489

 

Contrasting effects of different cannabinoid receptor ligands on mouse ingestive behavior (abst – 2012)  http://www.unboundmedicine.com/medline/ebm/record/22772336/abstract/Contrasting_effects_of_differen t_cannabinoid_receptor_ligands_on_mouse_ingestive_behaviour_

 

CB1 Agonist ACEA Protects Neurons and Reduces the Cognitive Impairment of AβPP/PS1 Mice.         (abst – 2012)                                  http://www.ncbi.nlm.nih.gov/pubmed/22451318

 

Protective effect of cannabinoid CB1 receptor activation against altered intrinsic repetitive firing properties induced by Aβ neurotoxicity.                                                                      (abst – 2012)  http://www.ncbi.nlm.nih.gov/pubmed/22172925

 

CB1 cannabinoid receptor activation rescues amyloid β-induced alterations in behaviour and intrinsic electrophysiological properties of rat hippocampal CA1 pyramidal neurones. (abst – 2012)                                    http://www.ncbi.nlm.nih.gov/pubmed/22508047

 

Opposing Roles for Cannabinoid Receptor Type-1 (CB(1)) and Transient Receptor Potential Vanilloid Type-1 Channel (TRPV1) on the Modulation of Panic-Like Responses in Rats.      (abst – 2012)                                            http://www.ncbi.nlm.nih.gov/pubmed/21937980

 

Contrasting protective effects of cannabinoids against oxidative stress and amyloid-β evoked neurotoxicity in vitro.                                                           (abst – 2012)      http://www.ncbi.nlm.nih.gov/pubmed/22233683

 

Cannabinoids and muscular pain. Effectiveness of the local administration in rat. (abst – 2012)                                   http://www.ncbi.nlm.nih.gov/pubmed/22354705

 

Revisiting CB1 Receptor as Drug Target in Human Melanoma.              (abst – 2012)

http://www.ncbi.nlm.nih.gov/pubmed/22447182

 

Photoperiodic Changes in Endocannabinoid Levels and Energetic Responses to Altered Signalling at CB1 Receptors in Siberian Hamsters                                               (abst – 2012)  http://onlinelibrary.wiley.com/doi/10.1111/j.1365-2826.2012.02312.x/abstract

 

Effect of ACEA-a selective cannabinoid CB1 receptor agonist on the protective action of different antiepileptic drugs in the mouse pentylenetetrazole-induced seizure model. (abst – 2012)                                       http://www.ncbi.nlm.nih.gov/pubmed/22789660

 

Evaluation of Anti-invasion Effect of Cannabinoids on Human Hepatocarcinoma Cells.

 

(abst – 2012)                       http://www.ncbi.nlm.nih.gov/pubmed/22978792

 

Distribution and function of the endocannabinoid system in the rat and human bladder. (abst – 2012)                                           http://www.ncbi.nlm.nih.gov/pubmed/23081739

 

Chronic activation of cannabinoid receptors in vitro does not compromise mouse islet function.   (abst – 2012)                                  http://www.ncbi.nlm.nih.gov/pubmed/23078523

 

Revisiting CB1 receptor as drug target in human melanoma.                      (abst – 2012)

http://www.ncbi.nlm.nih.gov/pubmed/22447182

 

Anti-Cancer Effects In Human Liver Cancer Cells Produced By Cannabis Agonists (news – 2012)                                           http://www.imarijuana.com/tag/cannabinoid-agonists

 

Type-1 (CB(1)) Cannabinoid Receptor Promotes Neuronal Differentiation and Maturation of Neural Stem Cells.                                                                            (abst – 2013)  http://www.ncbi.nlm.nih.gov/pubmed/23372698

 

Evaluation of anti-invasion effect of cannabinoids on human hepatocarcinoma cells. (abst – 2013)                                           http://www.ncbi.nlm.nih.gov/pubmed/22978792

 

Role of cannabinoid and vanilloid receptors in invasion of human breast carcinoma cells (abst – 2013)                                             http://www.ncbi.nlm.nih.gov/pubmed/23394450

 

 

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